Abstract
A new class of azabicyclo[3.1.0]benzenesulfonamides is presented as selective dopamine D3 antagonists together with SAR and selectivity data.
Copyright (c) 2010 Elsevier Ltd. All rights reserved.
MeSH terms
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Benzene / chemistry
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Benzene / pharmacology
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Dopamine Antagonists / chemistry*
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Dopamine Antagonists / pharmacology*
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Humans
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Receptors, Dopamine D3 / antagonists & inhibitors*
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Receptors, Dopamine D3 / metabolism*
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Structure-Activity Relationship
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Sulfonamides / chemistry*
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Sulfonamides / pharmacology*
Substances
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Dopamine Antagonists
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Receptors, Dopamine D3
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Sulfonamides
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Benzene